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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T6835 | Fenoldopam mesylate | Fenoldopam methanesulfonate,SKF-82526 mesylate,Corlopam mesylate,mesylate,SKF 82526 | Dopamine Receptor |
Fenoldopam mesylate (Corlopam mesylate) is a selective dopamine-1 receptor (DA1) agonist with natriuretic/diuretic properties. It lowers blood pressure through arteriolar vasodilation. | |||
T8044 | Ajmalicine | Lamuran,Delta-Yohimbine,Raubasine,Ajmalicin | Adrenergic Receptor |
Ajmalicine (Raubasine) (Raubasine) is a potent adrenolytic agent which preferentially blocks α1-adrenoceptor. Ajmalicine is an reversible but non-competitive nicotine receptor full inhibitor, IC50 = 72.3 μM. Ajmalicine a... | |||
TN1065 | Hirsutine | Apoptosis | |
Hirsutine induces apoptosis and is a potent Dengue virus inhibitor exhibiting low cytotoxicity.Hirsutine has anticancer, cardioprotective, anti-hypertensive and anti-arrhythmic activities, it also has vasodilatation acti... | |||
TCS1704 | Artemitin | Artemetin,Artemisetin,Erianthin | Antioxidant |
1. Artemitin (Erianthin) has anti-inflammatory activity. 2. Artemitin (Erianthin) protects endothelial function by acting as antioxidant and antiapoptotic agent and through the activation of ERK1/2 and Akt. 3. Intravenou... | |||
T21416 | Hydroflumethiazide | Diurometon,Glomerulin,Diuredemina,Flutizide,Hidroflumetiazid | |
Hydroflumethiazide is a thiazide diuretic. It has also shown the activity of anti-hypertensive. | |||
T17112 | Todralazine | Ecarazine | Others |
Todralazine is an anti-hypertensive agent and acts as a β2AR blocker. It also has an antioxidant and free radical scavenging activity. | |||
T15680 | L-159282 | MK 996 | Others |
L-159282 is an orally active and nonpeptide angiotensin II receptor antagonist. It also has anti-hypertensive activity. | |||
T62618 | SPH3127 | ||
SPH3127 (DRI 18) is a potent, orally active, novel direct renin inhibitor with IC50 values of 0.4 nM and 0.45 nM for recombinant human-renin and human plasma renin activity, respectively. SPH3127 has an anti-hypertensive... | |||
T69254 | Ajmalicine hydrochloride | Raubasine hydrochloride | |
Ajmalicine (Raubasine) hydrochloride, a potent adrenolytic compound, selectively inhibits α1-adrenoceptors and acts as a reversible, non-competitive full inhibitor of nicotine receptors with an IC50 of 72.3 μM. This chem... | |||
T62543 | JNc-440 | ||
JNc-440 is a potent anti-hypertensive agent. jNc-440 enhances the interaction between the transient receptor potential vanilloid subtype 4 (TRPV4) and calcium-activated potassium channel 3 (KCa2.3) in endothelial cells. ... |